Allosteric enhancers at the adenosine A1 receptor have received attention as anti-arrhythmic cardiac agents, and, more recently, as anti-lipolytic agents. In addn., allosteric modulators at the adenosine A1 receptor have therapeutic potential as analgesics and neuroprotective agents. In particular, the compds. with improved potency as enhancers and reduced antagonist properties are mentioned.
Allosteric enhancers for A(1) adenosine receptor
BARALDI, Pier Giovanni;IACONINOTO, Antonietta;PRETI, Delia;FRUTTAROLO, Francesca;AGHAZADEH TABRIZI, Mojgan;ROMAGNOLI, Romeo
2007
Abstract
Allosteric enhancers at the adenosine A1 receptor have received attention as anti-arrhythmic cardiac agents, and, more recently, as anti-lipolytic agents. In addn., allosteric modulators at the adenosine A1 receptor have therapeutic potential as analgesics and neuroprotective agents. In particular, the compds. with improved potency as enhancers and reduced antagonist properties are mentioned.File in questo prodotto:
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