PACIFICO, Salvatore
PACIFICO, Salvatore
Dipartimento di Scienze chimiche, farmaceutiche ed agrarie
A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism
2017 Fantinati, Anna; Bianco, Sara; Salvadori, Severo; Pacifico, Salvatore; Guerrini, Remo; Cerlesi, Maria Camilla; Trapella, Claudio; Calo', Girolamo
A Peptidic Thymidylate-Synthase Inhibitor Loaded on Pegylated Liposomes Enhances the Antitumour Effect of Chemotherapy Drugs in Human Ovarian Cancer Cells
2020 Marverti, Gaetano; Gozzi, Gaia; Maretti, Eleonora; Lauriola, Angela; Severi, Leda; Sacchetti, Francesca; Losi, Lorena; Pacifico, Salvatore; Ferrari, Stefania; Ponterini, Glauco; Leo, Eliana; Costi, Maria Paola; D'Arca, Domenico
Activation of nociceptin/orphanin FQ receptors inhibits contextual fear memory reconsolidation
file con accesso da definire2017 Rekik, Khaoula; Faria Da Silva, Raquel; Colom, Morgane; Pacifico, Salvatore; Zaveri, Nurulain T; Calo', Girolamo; Rampon, Claire; Frances, Bernard; Mouledous, Lionel
Age differentially impacts adaptive immune responses induced by adenoviral versus mRNA vaccines against COVID-19
2024 Dallan, Beatrice; Proietto, Davide; De Laurentis, Martina; Gallerani, Eleonora; Martino, Mara; Ghisellini, Sara; Zurlo, Amedeo; Volpato, Stefano; Govoni, Benedetta; Borghesi, Michela; Albanese, Valentina; Appay, Victor; Bonnini, Stefano; Llewellyn-Lacey, Sian; Pacifico, Salvatore; Grumiro, Laura; Brandolini, Martina; Semprini, Simona; Sambri, Vittorio; Ladell, Kristin; Parry, Helen M.; Moss, Paul A. H.; Price, David A.; Barbieri, Elena; Bernardi, Tatiana; Boni, Michela; Dall'Olio, Linda; De Laurentis, Martina; Fiorini, Caterina; Fiorini, Michele; Govoni, Maurizio; Neri, Margherita; Palma, Fabio; Romagnoni, Franco; Caputo, Antonella; Gavioli, Riccardo; Nicoli, Francesco
Age, Sex, Hypertension and HDL-C Alter Serum BACE1 Activity in Cognitively Normal Subjects: Implications for Alzheimer's Disease
2022 Cervellati, C; Vergallo, A; Trentini, A; Campo, G; Vieceli Dalla Sega, F; Bonaccorsi, G; Rosta, V; Renzini, C; Pacifico, S; Passaro, A; Hampel, H; Zuliani, G; Rizzo, P
Ageing Curtails the Diversity and Functionality of Nascent CD8+ T Cell Responses against SARS-CoV-2
2023 Proietto, Davide; Dallan, Beatrice; Gallerani, Eleonora; Albanese, Valentina; Llewellyn-Lacey, Sian; Price, David A.; Appay, Victor; Pacifico, Salvatore; Caputo, Antonella; Nicoli, Francesco; Gavioli, Riccardo
alpha-Diketones as acyl anion equivalents: a non-enzymatic thiamine-promoted route to aldehyde ketone coupling in PEG(400) as recyclable medium
file con accesso da definire2011 Bortolini, Olga; Fantin, Giancarlo; Fogagnolo, Marco; Giovannini, Pier Paolo; Venturi, Valentina; Pacifico, Salvatore; Massi, Alessandro
alpha-Diketones as acyl anion equivalents: new enzymatic and non-enzymatic thiamine-promoted routes to aldehyde-ketone coupling
file con accesso da definire2011 Bortolini, Olga; Fantin, Giancarlo; Fogagnolo, Marco; Giovannini, Pier Paolo; Venturi, Valentina; Massi, Alessandro; Pacifico, Salvatore
Biased Agonism at Nociceptin/Orphanin FQ Receptors: A Structure Activity Study on N/OFQ(1-13)-NH2
2020 Pacifico, S.; Ferrari, F.; Albanese, V.; Marzola, E.; Neto, J. A.; Ruzza, C.; Calo, G.; Preti, D.; Guerrini, R.
Bifunctional octadentate pseudopeptides as Zirconium-89 chelators for immuno-PET applications
2024 Albanese, Valentina; Roccatello, Chiara; Pacifico, Salvatore; Guerrini, Remo; Preti, Delia; Gentili, Silvia; Tegoni, Matteo; Remelli, Maurizio; Bellotti, Denise; Amico, Jonathan; Gorgoni, Giancarlo; Cazzola, Emiliano
COMPOSTI PIRROLIDINICI E PIPERIDINICI COME INIBITORI DELL’INFLAMMASOMA NLRP3 E LORO USO COME MEDICAMENTI
file con accesso da definire2022 Pinton, Paolo; Giorgi, Carlotta; Preti, Delia; Missiroli, Sonia; Albanese, Valentina; Pacifico, Salvatore
COMPOSTI SOLFONAMMIDICI COME INIBITORI DELL’INFLAMMASOMA NLRP3 E LORO USO COME MEDICAMENTI
file con accesso da definire2022 Pinton, Paolo; Giorgi, Carlotta; Preti, Delia; Missiroli, Sonia; Marisole, Perrone; Pacifico, Salvatore; Albanese, Valentina
COMPOSTI TETRAIDROISOCHINOLINICI COME INIBITORI DELL’INFLAMMASOMA NLRP3 E LORO USO COME MEDICAMENTI
file con accesso da definire2022 Pinton, Paolo; Giorgi, Carlotta; Preti, Delia; Missiroli, Sonia; Pacifico, Salvatore; Albanese, Valentina
Compounds as nlrp3 inflammasome inhibitors and their use as medicaments
file con accesso da definire2023 Pinton, Paolo; Giorgi, Carlotta; Preti, Delia; Pacifico, Salvatore; Perrone, Mariasole; Missiroli, Sonia; Albanese, Valentina.
Conformational Propensity and Biological Studies of Proline Mutated LR Peptides Inhibiting Human Thymidylate Synthase and Ovarian Cancer Cell Growth
2018 Saxena, P; Severi, L; Santucci, M; Taddia, L; Ferrari, S; Luciani, R; Marverti, G; Marraccini, C; Tondi, D; Mor, M; Scalvini, L; Vitiello, S; Losi, L; Fonda, S; Pacifico, S; Guerrini, R; D'Arca, D; Ponterini, G; Costi, Mp
Conveying a newly designed hydrophilic anti-human thymidylate synthase peptide to cisplatin resistant cancer cells: are pH-sensitive liposomes more effective than conventional ones?
file con accesso da definire2017 Sacchetti, Francesca; D'Arca, Domenico; Genovese, Filippo; Pacifico, Salvatore; Maretti, E; Hanuskova, M; Iannuccelli, V; Costi, Mp; Leo, E.
Cyclic peptides acting as allosteric inhibitors of human thymidylate synthase and cancer cell growth
2019 Pacifico, S.; Santucci, M.; Luciani, R.; Saxena, P.; Linciano, P.; Ponterini, G.; Lauriola, A.; D'Arca, D.; Marverti, G.; Guerrini, R.; Costi, M. P.
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones
2016 Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, Anna; Manfredini, Stefano; Pacifico, Salvatore; Liekens, Sandra; Balzarini, Jan
Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth
2022 Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; H Salo-Ahen, Outi M; Carosati, Emanuele; Franchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; Cardinale, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Gaetana Moschella, Maria; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; da Silva Cordeiro, Anabela; Giovannetti, Elisa; J Peters, Godefridus; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; M Stroud, Robert; C Wade, Rebecca; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Paola Costi, Maria
Dimethyl Sulfoxide and N,N-dimethylformamide as Umpolung Pre-catalysts in Cross Benzoin Reactions of alpha-Diketones with Aldehydes
file con accesso da definire2013 Bortolini, Olga; Massi, Alessandro; Giovannini, Pier Paolo; Pacifico, Salvatore; Ragno, Daniele; Zaghi, Anna
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism | 2017 | Fantinati, Anna; Bianco, Sara; Salvadori, Severo; Pacifico, Salvatore; Guerrini, Remo; Cerlesi, M... espandi | |
A Peptidic Thymidylate-Synthase Inhibitor Loaded on Pegylated Liposomes Enhances the Antitumour Effect of Chemotherapy Drugs in Human Ovarian Cancer Cells | 2020 | Marverti, Gaetano; Gozzi, Gaia; Maretti, Eleonora; Lauriola, Angela; Severi, Leda; Sacchetti, Fra... espandi | |
Activation of nociceptin/orphanin FQ receptors inhibits contextual fear memory reconsolidation | 2017 | Rekik, Khaoula; Faria Da Silva, Raquel; Colom, Morgane; Pacifico, Salvatore; Zaveri, Nurulain T; ... espandi | file con accesso da definire |
Age differentially impacts adaptive immune responses induced by adenoviral versus mRNA vaccines against COVID-19 | 2024 | Dallan, Beatrice; Proietto, Davide; De Laurentis, Martina; Gallerani, Eleonora; Martino, Mara; Gh... espandi | |
Age, Sex, Hypertension and HDL-C Alter Serum BACE1 Activity in Cognitively Normal Subjects: Implications for Alzheimer's Disease | 2022 | Cervellati, C; Vergallo, A; Trentini, A; Campo, G; Vieceli Dalla Sega, F; Bonaccorsi, G; Rosta, V... espandi | |
Ageing Curtails the Diversity and Functionality of Nascent CD8+ T Cell Responses against SARS-CoV-2 | 2023 | Proietto, Davide; Dallan, Beatrice; Gallerani, Eleonora; Albanese, Valentina; Llewellyn-Lacey, Si... espandi | |
alpha-Diketones as acyl anion equivalents: a non-enzymatic thiamine-promoted route to aldehyde ketone coupling in PEG(400) as recyclable medium | 2011 | Bortolini, Olga; Fantin, Giancarlo; Fogagnolo, Marco; Giovannini, Pier Paolo; Venturi, Valentina;... espandi | file con accesso da definire |
alpha-Diketones as acyl anion equivalents: new enzymatic and non-enzymatic thiamine-promoted routes to aldehyde-ketone coupling | 2011 | Bortolini, Olga; Fantin, Giancarlo; Fogagnolo, Marco; Giovannini, Pier Paolo; Venturi, Valentina;... espandi | file con accesso da definire |
Biased Agonism at Nociceptin/Orphanin FQ Receptors: A Structure Activity Study on N/OFQ(1-13)-NH2 | 2020 | Pacifico, S.; Ferrari, F.; Albanese, V.; Marzola, E.; Neto, J. A.; Ruzza, C.; Calo, G.; Preti, D.... espandi | |
Bifunctional octadentate pseudopeptides as Zirconium-89 chelators for immuno-PET applications | 2024 | Albanese, Valentina; Roccatello, Chiara; Pacifico, Salvatore; Guerrini, Remo; Preti, Delia; Genti... espandi | |
COMPOSTI PIRROLIDINICI E PIPERIDINICI COME INIBITORI DELL’INFLAMMASOMA NLRP3 E LORO USO COME MEDICAMENTI | 2022 | Pinton, Paolo; Giorgi, Carlotta; Preti, Delia; Missiroli, Sonia; Albanese, Valentina; Pacifico, S... espandi | file con accesso da definire |
COMPOSTI SOLFONAMMIDICI COME INIBITORI DELL’INFLAMMASOMA NLRP3 E LORO USO COME MEDICAMENTI | 2022 | Pinton, Paolo; Giorgi, Carlotta; Preti, Delia; Missiroli, Sonia; Marisole, Perrone; Pacifico, Sal... espandi | file con accesso da definire |
COMPOSTI TETRAIDROISOCHINOLINICI COME INIBITORI DELL’INFLAMMASOMA NLRP3 E LORO USO COME MEDICAMENTI | 2022 | Pinton, Paolo; Giorgi, Carlotta; Preti, Delia; Missiroli, Sonia; Pacifico, Salvatore; Albanese, V... espandi | file con accesso da definire |
Compounds as nlrp3 inflammasome inhibitors and their use as medicaments | 2023 | Pinton, Paolo; Giorgi, Carlotta; Preti, Delia; Pacifico, Salvatore; Perrone, Mariasole; Missiroli... espandi | file con accesso da definire |
Conformational Propensity and Biological Studies of Proline Mutated LR Peptides Inhibiting Human Thymidylate Synthase and Ovarian Cancer Cell Growth | 2018 | Saxena, P; Severi, L; Santucci, M; Taddia, L; Ferrari, S; Luciani, R; Marverti, G; Marraccini, C;... espandi | |
Conveying a newly designed hydrophilic anti-human thymidylate synthase peptide to cisplatin resistant cancer cells: are pH-sensitive liposomes more effective than conventional ones? | 2017 | Sacchetti, Francesca; D'Arca, Domenico; Genovese, Filippo; Pacifico, Salvatore; Maretti, E; Hanus... espandi | file con accesso da definire |
Cyclic peptides acting as allosteric inhibitors of human thymidylate synthase and cancer cell growth | 2019 | Pacifico, S.; Santucci, M.; Luciani, R.; Saxena, P.; Linciano, P.; Ponterini, G.; Lauriola, A.; D... espandi | |
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones | 2016 | Onnis, Valentina; Demurtas, Monica; Deplano, Alessandro; Balboni, Gianfranco; Baldisserotto, Anna... espandi | |
Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth | 2022 | Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; H Salo-Ahen, Outi M; Carosati, Emanuele; F... espandi | |
Dimethyl Sulfoxide and N,N-dimethylformamide as Umpolung Pre-catalysts in Cross Benzoin Reactions of alpha-Diketones with Aldehydes | 2013 | Bortolini, Olga; Massi, Alessandro; Giovannini, Pier Paolo; Pacifico, Salvatore; Ragno, Daniele; ... espandi | file con accesso da definire |