BARALDI, Stefania
BARALDI, Stefania
Dipartimento di Scienze Chimiche e Farmaceutiche (attivo dal 01/01/2012 al 31/12/2022)
1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists
file con accesso da definire2008 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Preti, Delia; Romagnoli, Romeo; Saponaro, Giulia; Baraldi, Stefania; Moorman, A. R.; Zaid, A. N.; Varani, Katia; Borea, Pier Andrea
2-Alkoxycarbonyl-3-arylamino-5-substituted thiophenes as a novel class of antimicrotubule agents: Design, synthesis, cell growth and tubulin polymerization inhibition
2018 Romagnoli, Romeo; Kimatrai Salvador, Maria; Schiaffino Ortega, Santiago; Baraldi, Pier Giovanni; Oliva, Paola; Baraldi, Stefania; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Balzarini, Jan; Liekens, Sandra; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro
3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization
2018 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists
2012 Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan
7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation
2012 Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; P., Pedretti; C., Fusi; R., Nassini; S., Materazzi; P., Geppetti; Preti, Delia
A 2a adenosine receptor: Structures, modeling, and medicinal chemistry
2018 Baraldi, S.; Baraldi, P. G.; Oliva, P.; Toti, K. S.; Ciancetta, A.; Jacobson, K. A.
A3 adenosine receptor antagonists: History and future perspectives
file con accesso da definire2010 Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; Baraldi, Stefania; Tabrizi, Mojgan Aghazadeh; Preti, Delia
A3 Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy
2018 Jacobson, Ka; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea; Baraldi, Stefania; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Baraldi, Pier Giovanni; Ciancetta, A; Tosh, Dk; Gao, Zg; Gessi, Stefania
Adenosine Receptors in Colon Carcinoma Tissues and Colon Tumoral Cell Lines: Focus on the A3 Adenosine Subtype
file con accesso da definire2007 Gessi, Stefania; Merighi, Stefania; Varani, Katia; Cattabriga, Elena; Benini, Annalisa; Mirandola, Prisco; E., Leung; S., MAC LENNAN; Feo, Carlo; Baraldi, Stefania; Borea, Pier Andrea
Design and Synthesis of New A2B Adenosine Receptor Antagonists
2009 Baraldi, Stefania
Design and Synthesis of Potent in Vitro and in Vivo Anticancer Agents Based on 1-(3’,4’,5’-Trimethoxyphenyl)-2-Aryl-1H-Imidazole
2016 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; AGHAZADEH TABRIZI, Mojgan; Lopez Cara, Carlota; Ferla, Salvatore; Brancale, Andrea; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Basso, Giuseppe; Viola, Giampietro .
Design, synthesis and biological evaluation of 3-substituted-2-oxindole hybrid derivatives as novel anticancer agents
2017 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Salvador, Maria Kimatrai; Lopez Cara, Luisa Carlota; Bortolozzi, Roberta; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro
Design, Synthesis, and Biological Evaluation of 6-Substituted Thieno[3,2-d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors
2019 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Schiaffino Ortega, Santiago; Chayah, Mariem; Kimatrai Salvador, Maria; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Mattiuzzo, Elena; Viola, Giampietro
Design, synthesis, and biological evaluation of novel 2-((2-(4-(substituted)phenylpiperazin-1-yl)ethyl)amino)-5'-N-ethylcarboxamidoadenosines as potent and selective agonists of the A2A adenosine receptor
2015 Preti, Delia; Baraldi, Pier Giovanni; Saponaro, Giulia; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; Cosconati, Sandro; Bruno, Agostino; Novellino, Ettore; Vincenzi, Fabrizio; Ravani, Annalisa; Borea, Pier Andrea; Varani, Katia
Design, Synthesis, and Pharmacological Properties of New Heteroarylpyridine/Heteroarylpyrimidine Derivatives as CB2 Cannabinoid Receptor Partial Agonists
file con accesso da definire2013 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Corciulo, Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors
2018 Aghazadeh Tabrizi, M.; Baraldi, P. G.; Baraldi, S.; Ruggiero, E.; De Stefano, L.; Rizzolio, F.; Di Cesare Mannelli, L.; Ghelardini, C.; Chicca, A.; Lapillo, M.; Gertsch, J.; Manera, C.; Macchia, M.; Martinelli, A.; Granchi, C.; Minutolo, F.; Tuccinardi, T.
Discovery of 7-oxopyrazolo[1,5-a]pyrimidine-6-carboxamides as potent and selective CB(2) cannabinoid receptor inverse agonists.
file con accesso da definire2013 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; Moorman, Ar; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Tintori, C; Tuccinardi, T; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Medicinal Chemistry, Pharmacology, and Clinical Implications of TRPV1 Receptor Antagonists
2017 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea
N-6-[(Hetero)aryl/(cyclo)alkyl-carbamoyi-methoxy-phenyl]-(2chloro)-5 '-N-ethylearboxamido-adenosines: The first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptor
file con accesso da definire2007 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Saponaro, Giulia; Baraldi, Stefania; Romagnoli, Romeo; Moorman, Ar; Gessi, Stefania; Varani, Katia; Borea, Pier Andrea
New 2-heterocyclyl-imidazo[2,1- i ]purin-5-one derivatives as potent and selective human A 3 adenosine receptor antagonists
file con accesso da definire2011 Baraldi, Pier Giovanni; Preti, Delia; Zaid, Na; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; Romagnoli, Romeo; Moorman, Ar; Varani, Katia; Cosconati, S; Di Maro, S; Marinelli, L; Novellino, E; Borea, Pier Andrea
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists | 2008 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Preti, Delia; Romagnoli, Romeo; Saponaro, Giul...ia; Baraldi, Stefania; Moorman, A. R.; Zaid, A. N.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| 2-Alkoxycarbonyl-3-arylamino-5-substituted thiophenes as a novel class of antimicrotubule agents: Design, synthesis, cell growth and tubulin polymerization inhibition | 2018 | Romagnoli, Romeo; Kimatrai Salvador, Maria; Schiaffino Ortega, Santiago; Baraldi, Pier Giovanni; ...Oliva, Paola; Baraldi, Stefania; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Balzarini, Jan; Liekens, Sandra; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro | |
| 3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization | 2018 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Bra...ncale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro | |
| 7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists | 2012 | Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi..., Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan | |
| 7-Substituted-pyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as antagonists of the transient receptor potential ankyrin 1 (TRPA1) channel: A promising approach for treating pain and inflammation | 2012 | Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Baraldi, S...tefania; P., Pedretti; C., Fusi; R., Nassini; S., Materazzi; P., Geppetti; Preti, Delia | |
| A 2a adenosine receptor: Structures, modeling, and medicinal chemistry | 2018 | Baraldi, S.; Baraldi, P. G.; Oliva, P.; Toti, K. S.; Ciancetta, A.; Jacobson, K. A. | |
| A3 adenosine receptor antagonists: History and future perspectives | 2010 | Baraldi, Pier Giovanni; Romagnoli, Romeo; Saponaro, Giulia; Baraldi, Stefania; Tabrizi, Mojgan Ag...hazadeh; Preti, Delia | file con accesso da definire |
| A3 Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy | 2018 | Jacobson, Ka; Merighi, Stefania; Varani, Katia; Borea, Pier Andrea; Baraldi, Stefania; AGHAZADEH ...TABRIZI, Mojgan; Romagnoli, Romeo; Baraldi, Pier Giovanni; Ciancetta, A; Tosh, Dk; Gao, Zg; Gessi, Stefania | |
| Adenosine Receptors in Colon Carcinoma Tissues and Colon Tumoral Cell Lines: Focus on the A3 Adenosine Subtype | 2007 | Gessi, Stefania; Merighi, Stefania; Varani, Katia; Cattabriga, Elena; Benini, Annalisa; Mirandola..., Prisco; E., Leung; S., MAC LENNAN; Feo, Carlo; Baraldi, Stefania; Borea, Pier Andrea | file con accesso da definire |
| Design and Synthesis of New A2B Adenosine Receptor Antagonists | 2009 | Baraldi, Stefania | |
| Design and Synthesis of Potent in Vitro and in Vivo Anticancer Agents Based on 1-(3’,4’,5’-Trimethoxyphenyl)-2-Aryl-1H-Imidazole | 2016 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; AGH...AZADEH TABRIZI, Mojgan; Lopez Cara, Carlota; Ferla, Salvatore; Brancale, Andrea; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Basso, Giuseppe; Viola, Giampietro . | |
| Design, synthesis and biological evaluation of 3-substituted-2-oxindole hybrid derivatives as novel anticancer agents | 2017 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Sal...vador, Maria Kimatrai; Lopez Cara, Luisa Carlota; Bortolozzi, Roberta; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro | |
| Design, Synthesis, and Biological Evaluation of 6-Substituted Thieno[3,2-d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors | 2019 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Sch...iaffino Ortega, Santiago; Chayah, Mariem; Kimatrai Salvador, Maria; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Mattiuzzo, Elena; Viola, Giampietro | |
| Design, synthesis, and biological evaluation of novel 2-((2-(4-(substituted)phenylpiperazin-1-yl)ethyl)amino)-5'-N-ethylcarboxamidoadenosines as potent and selective agonists of the A2A adenosine receptor | 2015 | Preti, Delia; Baraldi, Pier Giovanni; Saponaro, Giulia; Romagnoli, Romeo; AGHAZADEH TABRIZI, Mojg...an; Baraldi, Stefania; Cosconati, Sandro; Bruno, Agostino; Novellino, Ettore; Vincenzi, Fabrizio; Ravani, Annalisa; Borea, Pier Andrea; Varani, Katia | |
| Design, Synthesis, and Pharmacological Properties of New Heteroarylpyridine/Heteroarylpyrimidine Derivatives as CB2 Cannabinoid Receptor Partial Agonists | 2013 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, R...omeo; Preti, Delia; Baraldi, Stefania; Corciulo, Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
| Discovery of 1,5-Diphenylpyrazole-3-Carboxamide Derivatives as Potent, Reversible, and Selective Monoacylglycerol Lipase (MAGL) Inhibitors | 2018 | Aghazadeh Tabrizi, M.; Baraldi, P. G.; Baraldi, S.; Ruggiero, E.; De Stefano, L.; Rizzolio, F.; D...i Cesare Mannelli, L.; Ghelardini, C.; Chicca, A.; Lapillo, M.; Gertsch, J.; Manera, C.; Macchia, M.; Martinelli, A.; Granchi, C.; Minutolo, F.; Tuccinardi, T. | |
| Discovery of 7-oxopyrazolo[1,5-a]pyrimidine-6-carboxamides as potent and selective CB(2) cannabinoid receptor inverse agonists. | 2013 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Saponaro, Giulia; Moorman, Ar; Romagnoli, Rome...o; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Tintori, C; Tuccinardi, T; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
| Medicinal Chemistry, Pharmacology, and Clinical Implications of TRPV1 Receptor Antagonists | 2017 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Gessi, Stefania; Merighi, S...tefania; Borea, Pier Andrea | |
| N-6-[(Hetero)aryl/(cyclo)alkyl-carbamoyi-methoxy-phenyl]-(2chloro)-5 '-N-ethylearboxamido-adenosines: The first example of adenosine-related structures with potent agonist activity at the human A(2B) adenosine receptor | 2007 | Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Saponaro,... Giulia; Baraldi, Stefania; Romagnoli, Romeo; Moorman, Ar; Gessi, Stefania; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| New 2-heterocyclyl-imidazo[2,1- i ]purin-5-one derivatives as potent and selective human A 3 adenosine receptor antagonists | 2011 | Baraldi, Pier Giovanni; Preti, Delia; Zaid, Na; Saponaro, Giulia; AGHAZADEH TABRIZI, Mojgan; Bara...ldi, Stefania; Romagnoli, Romeo; Moorman, Ar; Varani, Katia; Cosconati, S; Di Maro, S; Marinelli, L; Novellino, E; Borea, Pier Andrea | file con accesso da definire |