VARANI, Katia
VARANI, Katia
Dipartimento di Medicina Traslazionale e per la Romagna
1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists
file con accesso da definire2008 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Preti, Delia; Romagnoli, Romeo; Saponaro, Giulia; Baraldi, Stefania; Moorman, A. R.; Zaid, A. N.; Varani, Katia; Borea, Pier Andrea
1-Methyl and 1-(2-hydroxyalkyl)-5-(3-alkyl/cycloalkyl/phenyl/naphthylureido)-1H-pyrazole-4-carboxylic acid ethyl esters as potent human neutrophil chemotaxis inhibitors
2009 Bruno, O; Brullo, C; Bondavalli, F; Schenone, S; Spisani, Susanna; Falzarano, Ms; Varani, Katia; Barocelli, E; Ballabeni, V; Giorgio, C; Tognolini, M.
1H-pyrazolo[4,3-d]pyrimidine-7(6H)-one and 5H-pyrazolo[4,3-d] 1,2,3-triazin-4(3H)-one derivatives. Synthesis and in vitro biological activity at adenosine A1 and A2a receptors
file con accesso da definire1996 Baraldi, Pier Giovanni; Cacciari, Barbara; Dalpiaz, Alessandro; Dionisotti, S.; Zocchi, C.; PINEDA DE LAS INFANTAS, M. J.; Spalluto, G.; Varani, Katia
2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators
file con accesso da definire2023 Oliva, Paola; Suresh, R Rama; Pasquini, Silvia; Salmaso, Veronica; Will, Edward J; Tosh, Dilip K; Gao, Zhan-Guo; Liu, Naili; Gavrilova, Oksana; Vincenzi, Fabrizio; Varani, Katia; Jacobson, Kenneth A
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors
2022 Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
2-arylpyrazolo[3,4-c]quinolin-4-heteroaroylamines as potent and selective human A3 adenosine receptor antagonists. Synthesis and biological evaluetion.
file con accesso da definire2006 Catarzi, D.; Colotta, V.; Varano, F.; Capelli, F.; Lenzi, O.; Varani, Katia
2-Arylpyrazolo[4,3-d]pyrimidin-7-amino derivatives as new potent and selective human A3 adenosine receptor antagonists. Molecular modeling studies and pharmacological evaluation
file con accesso da definire2013 Squarcialupi, L.; Colotta, V.; Catarzi, D.; Varano, F.; Filacchioni, G.; Varani, Katia; Corciulo, Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Ghelardini, C.; Di Cesare Mannelli, L.; Ciancetta, A.; Moro, S.
2-phenyl-2,3-dihydro-1H-imidazo[1,2-b]pyrozole derivatives: new potent inhibitors of fMLP-induced neutrophil chemotaxis
file con accesso da definire2007 Bruno, O; Brullo, C; Bondavalli, F; Ranise, A; Schenone, S; FALZARANO M., S; Varani, K; Spisani, S
2-Phenylpyrazolo[4,3-d]pyrimidin-7-one as a New Scaffold To Obtain Potent and Selective Human A(3) Adenosine Receptor Antagonists: New Insights into the Receptor-Antagonist Recognition (dagger).
file con accesso da definire2009 Lenzi, O.; Colotta, V.; Catarzi, D.; Varano, F.; Poli, D.; Filacchioni, G.; Varani, Katia; Vincenzi, Fabrizio; Borea, Pier Andrea; Paoletta, S.; Morizzo, E.; Moro, S.
3H SCH 58261 labelling of functional A2A adenosine receptors in human neutrophil membranes
file con accesso da definire1998 Varani, Katia; Gessi, Stefania; Dionisotti, S; Ongini, E; Borea, Pier Andrea
4-amido-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones as a new potent and selective human A3 adenosine receptor antagonists. Synthesis, pharmacological evaluation, and ligand-receptor modeling studies.
file con accesso da definire2006 Lenzi, O; Colotta, V; Catarzi, D; Varano, F; Filacchioni, G; Martini, C; Trincavelli, L; Ciampi, O; Varani, Katia; Marighetti, F; Morizzo, E; Moro, S.
4-Heteroaryl Substituted Amino-3,5-Dicyanopyridines as New Adenosine Receptor Ligands: Novel Insights on Structure-Activity Relationships and Perspectives
2022 Catarzi, D.; Varano, F.; Vigiani, E.; Calenda, S.; Melani, F.; Varani, K.; Vincenzi, F.; Pasquini, S.; Mennini, N.; Nerli, G.; Dal Ben, D.; Volpini, R.; Colotta, V.
5-heteroarylcarbamoylamino-pyrazolo-triazolo pyrimidines as hA3 adenosine receptor antagonists.
file con accesso da definire2006 Pastorin, G.; Da Ros, T.; Bolcato, C.; Montopoli, C.; Moro, S.; Cacciari, Barbara; Baraldi, Pier Giovanni; Varani, Katia; Borea, Pier Andrea; Spalluto, G.
6-Amino-2-mercapto-3H-pyrimidin-4-one derivatives as new candidates for the antagonism at the P2Y12 receptors
file con accesso da definire2009 Crepaldi, Pamela; Cacciari, Barbara; Bonache, M. C.; Spalluto, G.; Varani, Katia; Borea, Pier Andrea; Kügelgen, I.; Hoffmann, K.; Pugliano, M.; Razzari, C.; Cattaneo, M.
7-Amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives: Structural investigations at the 5-position to target human A(1) and A(2A) adenosine receptors. Molecular modeling and pharmacological studies
2014 Squarcialupi, L; Colotta, V; Catarzi, D; Varano, F; Betti, M; Varani, Katia; Vincenzi, Fabrizio; Borea, Pier Andrea; Porta, N; Ciancetta, A; Moro, S.
7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists
2012 Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi, Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan
7-sobstituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonist: importance of modifications at the side chain on the activity and solubility.
file con accesso da definire2001 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
7-substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A(2A) adenosine receptor antagonists: A study on the importance of modifications at the side chain on the activity and solubility
file con accesso da definire2002 Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
7-substituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: importance of modifications at the side chain on the activity and solubility.
file con accesso da definire2001 Cacciari, Barbara; Baraldi, Pier Giovanni; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; Ongini, E.; Varani, Katia; Borea, Pier Andrea
[3H] CGS 21680 binding to purified adenosine A2A receptors in human platelets
file con accesso da definire1996 Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonists | 2008 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Preti, Delia; Romagnoli, Romeo; Saponaro, Giul...ia; Baraldi, Stefania; Moorman, A. R.; Zaid, A. N.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| 1-Methyl and 1-(2-hydroxyalkyl)-5-(3-alkyl/cycloalkyl/phenyl/naphthylureido)-1H-pyrazole-4-carboxylic acid ethyl esters as potent human neutrophil chemotaxis inhibitors | 2009 | Bruno, O; Brullo, C; Bondavalli, F; Schenone, S; Spisani, Susanna; Falzarano, Ms; Varani, Katia; ...Barocelli, E; Ballabeni, V; Giorgio, C; Tognolini, M. | |
| 1H-pyrazolo[4,3-d]pyrimidine-7(6H)-one and 5H-pyrazolo[4,3-d] 1,2,3-triazin-4(3H)-one derivatives. Synthesis and in vitro biological activity at adenosine A1 and A2a receptors | 1996 | Baraldi, Pier Giovanni; Cacciari, Barbara; Dalpiaz, Alessandro; Dionisotti, S.; Zocchi, C.; PINED...A DE LAS INFANTAS, M. J.; Spalluto, G.; Varani, Katia | file con accesso da definire |
| 2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators | 2023 | Oliva, Paola; Suresh, R Rama; Pasquini, Silvia; Salmaso, Veronica; Will, Edward J; Tosh, Dilip K;... Gao, Zhan-Guo; Liu, Naili; Gavrilova, Oksana; Vincenzi, Fabrizio; Varani, Katia; Jacobson, Kenneth A | file con accesso da definire |
| 2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors | 2022 | Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Va...leria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto | |
| 2-arylpyrazolo[3,4-c]quinolin-4-heteroaroylamines as potent and selective human A3 adenosine receptor antagonists. Synthesis and biological evaluetion. | 2006 | Catarzi, D.; Colotta, V.; Varano, F.; Capelli, F.; Lenzi, O.; Varani, Katia | file con accesso da definire |
| 2-Arylpyrazolo[4,3-d]pyrimidin-7-amino derivatives as new potent and selective human A3 adenosine receptor antagonists. Molecular modeling studies and pharmacological evaluation | 2013 | Squarcialupi, L.; Colotta, V.; Catarzi, D.; Varano, F.; Filacchioni, G.; Varani, Katia; Corciulo,... Carmen; Vincenzi, Fabrizio; Borea, Pier Andrea; Ghelardini, C.; Di Cesare Mannelli, L.; Ciancetta, A.; Moro, S. | file con accesso da definire |
| 2-phenyl-2,3-dihydro-1H-imidazo[1,2-b]pyrozole derivatives: new potent inhibitors of fMLP-induced neutrophil chemotaxis | 2007 | Bruno, O; Brullo, C; Bondavalli, F; Ranise, A; Schenone, S; FALZARANO M., S; Varani, K; Spisani, S | file con accesso da definire |
| 2-Phenylpyrazolo[4,3-d]pyrimidin-7-one as a New Scaffold To Obtain Potent and Selective Human A(3) Adenosine Receptor Antagonists: New Insights into the Receptor-Antagonist Recognition (dagger). | 2009 | Lenzi, O.; Colotta, V.; Catarzi, D.; Varano, F.; Poli, D.; Filacchioni, G.; Varani, Katia; Vincen...zi, Fabrizio; Borea, Pier Andrea; Paoletta, S.; Morizzo, E.; Moro, S. | file con accesso da definire |
| 3H SCH 58261 labelling of functional A2A adenosine receptors in human neutrophil membranes | 1998 | Varani, Katia; Gessi, Stefania; Dionisotti, S; Ongini, E; Borea, Pier Andrea | file con accesso da definire |
| 4-amido-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones as a new potent and selective human A3 adenosine receptor antagonists. Synthesis, pharmacological evaluation, and ligand-receptor modeling studies. | 2006 | Lenzi, O; Colotta, V; Catarzi, D; Varano, F; Filacchioni, G; Martini, C; Trincavelli, L; Ciampi, ...O; Varani, Katia; Marighetti, F; Morizzo, E; Moro, S. | file con accesso da definire |
| 4-Heteroaryl Substituted Amino-3,5-Dicyanopyridines as New Adenosine Receptor Ligands: Novel Insights on Structure-Activity Relationships and Perspectives | 2022 | Catarzi, D.; Varano, F.; Vigiani, E.; Calenda, S.; Melani, F.; Varani, K.; Vincenzi, F.; Pasquini..., S.; Mennini, N.; Nerli, G.; Dal Ben, D.; Volpini, R.; Colotta, V. | |
| 5-heteroarylcarbamoylamino-pyrazolo-triazolo pyrimidines as hA3 adenosine receptor antagonists. | 2006 | Pastorin, G.; Da Ros, T.; Bolcato, C.; Montopoli, C.; Moro, S.; Cacciari, Barbara; Baraldi, Pier ...Giovanni; Varani, Katia; Borea, Pier Andrea; Spalluto, G. | file con accesso da definire |
| 6-Amino-2-mercapto-3H-pyrimidin-4-one derivatives as new candidates for the antagonism at the P2Y12 receptors | 2009 | Crepaldi, Pamela; Cacciari, Barbara; Bonache, M. C.; Spalluto, G.; Varani, Katia; Borea, Pier And...rea; Kügelgen, I.; Hoffmann, K.; Pugliano, M.; Razzari, C.; Cattaneo, M. | file con accesso da definire |
| 7-Amino-2-phenylpyrazolo[4,3-d]pyrimidine derivatives: Structural investigations at the 5-position to target human A(1) and A(2A) adenosine receptors. Molecular modeling and pharmacological studies | 2014 | Squarcialupi, L; Colotta, V; Catarzi, D; Varano, F; Betti, M; Varani, Katia; Vincenzi, Fabrizio; ...Borea, Pier Andrea; Porta, N; Ciancetta, A; Moro, S. | |
| 7-Oxo-[1,4]oxazino[2,3,4-ij]quinoline-6-carboxamides as Selective CB2 Cannabinoid Receptor Ligands: Structural Investigations around a Novel Class of Full Agonists | 2012 | Baraldi, Pier Giovanni; Saponaro, Giulia; A. R., Moorman; Romagnoli, Romeo; Preti, Delia; Baraldi..., Stefania; Ruggiero, Emanuela; Varani, Katia; Targa, Martina; Vincenzi, Fabrizio; Borea, Pier Andrea; AGHAZADEH TABRIZI, Mojgan | |
| 7-sobstituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonist: importance of modifications at the side chain on the activity and solubility. | 2001 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; O...ngini, E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| 7-substituted 5-amino-2-(2-furyl)pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidines as A(2A) adenosine receptor antagonists: A study on the importance of modifications at the side chain on the activity and solubility | 2002 | Baraldi, Pier Giovanni; Cacciari, Barbara; Romagnoli, Romeo; Spalluto, G.; Monopoli, A.; Ongini, ...E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| 7-substituted-5-amino-2-(furyl)-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines as A2A adenosine receptor antagonists: importance of modifications at the side chain on the activity and solubility. | 2001 | Cacciari, Barbara; Baraldi, Pier Giovanni; Romagnoli, Romeo; Spalluto, Giampiero; Monopoli, A.; O...ngini, E.; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
| [3H] CGS 21680 binding to purified adenosine A2A receptors in human platelets | 1996 | Varani, Katia; Gessi, Stefania; Dalpiaz, Alessandro; Ongini, E.; Borea, Pier Andrea | file con accesso da definire |