PRENCIPE, Filippo
PRENCIPE, Filippo
Dipartimento di Scienze Chimiche e Farmaceutiche (attivo dal 01/01/2012 al 31/12/2022)
3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization
2018 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro
Apoptosis Pathways Triggered by a Potent Antiproliferative Hybrid Chalcone on Human Melanoma Cells
2021 Rodríguez, Irene; Saavedra, Ester; del Rosario, Henoc; Perdomo, Juan; Quintana, José; Prencipe, Filippo; Oliva, Paola; Romagnoli, Romeo; Estévez, Francisco
Cinnamic acid derivatives linked to arylpiperazines as novel potent inhibitors of tyrosinase activity and melanin synthesis
2022 Romagnoli, Romeo; Oliva, Paola; Prencipe, Filippo; Manfredini, Stefano; Germanò, Maria Paola; De Luca, Laura; Ricci, Federico; Corallo, Diana; Aveic, Sanja; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta
Design and Synthesis of Potent in Vitro and in Vivo Anticancer Agents Based on 1-(3’,4’,5’-Trimethoxyphenyl)-2-Aryl-1H-Imidazole
2016 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; AGHAZADEH TABRIZI, Mojgan; Lopez Cara, Carlota; Ferla, Salvatore; Brancale, Andrea; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Basso, Giuseppe; Viola, Giampietro .
Design, synthesis and antiproliferative activity of novel heterobivalent hybrids based on imidazo[2,1-b][1,3,4]thiadiazole and imidazo[2,1-b][1,3]thiazole scaffolds
2015 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Balzarini, Jan; Liekens, Sandra; Estévez, Francisco
Design, synthesis and biological evaluation of 2-alkoxycarbonyl-3-anilinoindoles as a new class of potent inhibitors of tubulin polymerization
2020 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Kimatrai Salvador, Maria; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Viola, Giampietro; Bortolozzi, Roberta; Persoons, Leentje; Balzarini, Jan; Liekens, Sandra; Schols, Dominique
Design, synthesis and biological evaluation of 3-substituted-2-oxindole hybrid derivatives as novel anticancer agents
2017 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Salvador, Maria Kimatrai; Lopez Cara, Luisa Carlota; Bortolozzi, Roberta; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro
Design, Synthesis and Biological Evaluation of Arylcinnamide Hybrid Derivatives as Novel Anticancer Agents
file con accesso da definire2014 Romagnoli, Romeo; Baraldi, Pier Giovanni; Maria Kimatrai, Salvador; Mariem, Chayah; M., Encarnacion Camacho; Prencipe, Filippo; Ernest, Hamel; Francesca, Consolaro; Giuseppe, Basso; Giampietro, Viola
Design, Synthesis, and Biological Evaluation of 6-Substituted Thieno[3,2-d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors
2019 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Schiaffino Ortega, Santiago; Chayah, Mariem; Kimatrai Salvador, Maria; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Mattiuzzo, Elena; Viola, Giampietro
Design, synthesis, in vitro, and in vivo anticancer and antiangiogenic activity of novel 3-arylaminobenzofuran derivatives targeting the colchicine site on tubulin
2015 Romagnoli, Romeo; Baraldi, Pier Giovanni; Salvador, Maria Kimatrai; Prencipe, Filippo; Lopez Cara, Carlota; Schiaffino Ortega, Santiago; Brancale, Andrea; Hamel, Ernest; Castagliuolo, Ignazio; Mitola, Stefania; Ronca, Roberto; Bortolozzi, Roberta; Porcù, Elena; Basso, Giuseppe; Viola, Giampietro
Novel iodoacetamido benzoheterocyclic derivatives with potent antileukemic activity are inhibitors of STAT5 phosphorylation
2016 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Lopez Cara, Carlota; Rondanin, Riccardo; Simoni, Daniele; Hamel, Ernest; Grimaudo, Stefania; Pipitone, Rosaria Maria; Meli, Maria; Tolomeo, Manlio
Synthesis and biological evaluation in vitro and in vivo of novel potent anticancer agents affecting tubulin polymerization
2017 Prencipe, Filippo
Synthesis and Biological Evaluation of 2-Methyl-4,5-Disubstituted Oxazoles as a Novel Class of Highly Potent Antitubulin Agents
2017 Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Salvador, Maria Kimatrai; Lopez Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Porcù, Elena; Basso, Giuseppe; Viola, Giampietro
Synthesis and biological evaluation of alpha-bromoacryloylamido indolyl pyridinyl propenones as potent apoptotic inducers in human leukaemia cells
2018 Romagnoli, Romeo; Prencipe, Filippo; Lopez-Cara, Luisa Carlota; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Estévez-Sarmiento, Francisco; Quintana, José; Estévez, Francisco
Synthesis and biological evaluation of new antitubulin agents containing 2-(30,40,50-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold
2020 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sandra; Hamel, Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto
Synthesis and Biological Evaluation of Pyrazolo[3,4-b]pyridin-4-ones as a New Class of Topoisomerase II Inhibitors
file con accesso da definire2015 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Prencipe, Filippo; Preti, Delia; Saponaro, Giulia; Romagnoli, Romeo; Gessi, Stefania; Merighi, Stefania; Stefanelli, Angela; Fazzi, Debora; Borea, Pier Andrea; Maia, Rodolfo C. outo; Romeiro, Nelilma C.; Fraga, Carlos A. M; Barreiro, Eliezer J.
Synthesis, Antimitotic and Antivascular Activity of 1-(3’,4’,5’-Trimethoxybenzoyl)-3-Arylamino-5-Amino-1,2,4-Triazoles
file con accesso da definire2014 Romagnoli, Romeo; Baraldi, Pier Giovanni; Kimatrai Salvador, M.; Prencipe, Filippo; Bertolasi, Valerio; Cancellieri, M.; Brancale, A.; Hamel, E.; Castagliuolo, I.; Consolaro, F.; Porcù, E.; Basso, G.; Viola, G.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 3-Aryl/Heteroaryl-5-amino-1-(3′,4′,5′-trimethoxybenzoyl)-1,2,4-triazoles as antimicrotubule agents. Design, synthesis, antiproliferative activity and inhibition of tubulin polymerization | 2018 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Bra...ncale, Andrea; Ferla, Salvatore; Hamel, Ernest; Bortolozzi, Roberta; Viola, Giampietro | |
| Apoptosis Pathways Triggered by a Potent Antiproliferative Hybrid Chalcone on Human Melanoma Cells | 2021 | Rodríguez, Irene; Saavedra, Ester; del Rosario, Henoc; Perdomo, Juan; Quintana, José; Prencipe, F...ilippo; Oliva, Paola; Romagnoli, Romeo; Estévez, Francisco | |
| Cinnamic acid derivatives linked to arylpiperazines as novel potent inhibitors of tyrosinase activity and melanin synthesis | 2022 | Romagnoli, Romeo; Oliva, Paola; Prencipe, Filippo; Manfredini, Stefano; Germanò, Maria Paola; De ...Luca, Laura; Ricci, Federico; Corallo, Diana; Aveic, Sanja; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta | |
| Design and Synthesis of Potent in Vitro and in Vivo Anticancer Agents Based on 1-(3’,4’,5’-Trimethoxyphenyl)-2-Aryl-1H-Imidazole | 2016 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; AGH...AZADEH TABRIZI, Mojgan; Lopez Cara, Carlota; Ferla, Salvatore; Brancale, Andrea; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Basso, Giuseppe; Viola, Giampietro . | |
| Design, synthesis and antiproliferative activity of novel heterobivalent hybrids based on imidazo[2,1-b][1,3,4]thiadiazole and imidazo[2,1-b][1,3]thiazole scaffolds | 2015 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Balzarini, Jan; Liekens, Sandra; Est...évez, Francisco | |
| Design, synthesis and biological evaluation of 2-alkoxycarbonyl-3-anilinoindoles as a new class of potent inhibitors of tubulin polymerization | 2020 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Kimatrai Salvador, Maria; Brancale, Andrea; Fe...rla, Salvatore; Hamel, Ernest; Viola, Giampietro; Bortolozzi, Roberta; Persoons, Leentje; Balzarini, Jan; Liekens, Sandra; Schols, Dominique | |
| Design, synthesis and biological evaluation of 3-substituted-2-oxindole hybrid derivatives as novel anticancer agents | 2017 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Sal...vador, Maria Kimatrai; Lopez Cara, Luisa Carlota; Bortolozzi, Roberta; Mattiuzzo, Elena; Basso, Giuseppe; Viola, Giampietro | |
| Design, Synthesis and Biological Evaluation of Arylcinnamide Hybrid Derivatives as Novel Anticancer Agents | 2014 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Maria Kimatrai, Salvador; Mariem, Chayah; M., Encarnaci...on Camacho; Prencipe, Filippo; Ernest, Hamel; Francesca, Consolaro; Giuseppe, Basso; Giampietro, Viola | file con accesso da definire |
| Design, Synthesis, and Biological Evaluation of 6-Substituted Thieno[3,2-d]pyrimidine Analogues as Dual Epidermal Growth Factor Receptor Kinase and Microtubule Inhibitors | 2019 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Baraldi, Pier Giovanni; Sch...iaffino Ortega, Santiago; Chayah, Mariem; Kimatrai Salvador, Maria; Lopez-Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Mattiuzzo, Elena; Viola, Giampietro | |
| Design, synthesis, in vitro, and in vivo anticancer and antiangiogenic activity of novel 3-arylaminobenzofuran derivatives targeting the colchicine site on tubulin | 2015 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Salvador, Maria Kimatrai; Prencipe, Filippo; Lopez Cara..., Carlota; Schiaffino Ortega, Santiago; Brancale, Andrea; Hamel, Ernest; Castagliuolo, Ignazio; Mitola, Stefania; Ronca, Roberto; Bortolozzi, Roberta; Porcù, Elena; Basso, Giuseppe; Viola, Giampietro | |
| Novel iodoacetamido benzoheterocyclic derivatives with potent antileukemic activity are inhibitors of STAT5 phosphorylation | 2016 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Lopez Cara, Carlota; Rondanin, Ricca...rdo; Simoni, Daniele; Hamel, Ernest; Grimaudo, Stefania; Pipitone, Rosaria Maria; Meli, Maria; Tolomeo, Manlio | |
| Synthesis and biological evaluation in vitro and in vivo of novel potent anticancer agents affecting tubulin polymerization | 2017 | Prencipe, Filippo | |
| Synthesis and Biological Evaluation of 2-Methyl-4,5-Disubstituted Oxazoles as a Novel Class of Highly Potent Antitubulin Agents | 2017 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Oliva, Paola; Baraldi, Stefania; Sal...vador, Maria Kimatrai; Lopez Cara, Luisa Carlota; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Ronca, Roberto; Bortolozzi, Roberta; Mariotto, Elena; Porcù, Elena; Basso, Giuseppe; Viola, Giampietro | |
| Synthesis and biological evaluation of alpha-bromoacryloylamido indolyl pyridinyl propenones as potent apoptotic inducers in human leukaemia cells | 2018 | Romagnoli, Romeo; Prencipe, Filippo; Lopez-Cara, Luisa Carlota; Oliva, Paola; Baraldi, Stefania; ...Baraldi, Pier Giovanni; Estévez-Sarmiento, Francisco; Quintana, José; Estévez, Francisco | |
| Synthesis and biological evaluation of new antitubulin agents containing 2-(30,40,50-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold | 2020 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sa...ndra; Hamel, Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto | |
| Synthesis and Biological Evaluation of Pyrazolo[3,4-b]pyridin-4-ones as a New Class of Topoisomerase II Inhibitors | 2015 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Prencipe, Filippo; Preti, D...elia; Saponaro, Giulia; Romagnoli, Romeo; Gessi, Stefania; Merighi, Stefania; Stefanelli, Angela; Fazzi, Debora; Borea, Pier Andrea; Maia, Rodolfo C. outo; Romeiro, Nelilma C.; Fraga, Carlos A. M; Barreiro, Eliezer J. | file con accesso da definire |
| Synthesis, Antimitotic and Antivascular Activity of 1-(3’,4’,5’-Trimethoxybenzoyl)-3-Arylamino-5-Amino-1,2,4-Triazoles | 2014 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Kimatrai Salvador, M.; Prencipe, Filippo; Bertolasi, Va...lerio; Cancellieri, M.; Brancale, A.; Hamel, E.; Castagliuolo, I.; Consolaro, F.; Porcù, E.; Basso, G.; Viola, G. | file con accesso da definire |