Sfoglia per Titolo
Synthesis and Biological Evaluation of Diastereoisomerically Pure N,O-Nucleosides
file con accesso da definire2010 B., Russo; Bortolini, Olga; A., De Nino; A., Garofalo; A., Melicchio; L., Maiuolo
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity
2016 Di Capua, A; Sticozzi, Claudia; Brogi, S; Brindisi, M; Cappelli, A; Sautebin, L; Rossi, A; Pace, S; Ghelardini, C; Di Cesare Mannelli, L; Valacchi, Giuseppe; Giorgi, Giulia; Giordani, Alice; Poce, G; Biava, M; Anzini, M.
Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents
2022 Oliva, Paola; Romagnoli, Romeo; Cacciari, Barbara; Manfredini, Stefano; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Milan, Noemi; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta
Synthesis and biological evaluation of new 8-heterocyclic xanthine derivative as highly potent and selective human A2B adenosine receptor antagonist
file con accesso da definire2006 Baraldi, Pier Giovanni; Tabrizi, M. A.; Preti, Delia; Bovero, A.; Romagnoli, Romeo; Fruttarolo, Francesca; Zaid, N. A.; Moorman, A. R.; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea
Synthesis and biological evaluation of new active For-Met-Leu-Phe-OMe analogues containing para-substituted Phe residues. J.Pept.Sci, 18, 418-426, 2012.
file con accesso da definire2012 Mollica, A.; Feliciani, F.; Stefanucci, A.; Costante, R.; Lucente, G.; Pinnen, F.; Notaristefano, D.; Spisani, Susanna
Synthesis and biological evaluation of new antitubulin agents containing 2-(30,40,50-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold
2020 Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sandra; Hamel, Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto
Synthesis and biological evaluation of new vinyl ester pseudotripeptide proteasome inhibitors
file con accesso da definire2006 Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]-9H-purin-9-yl]-N-ethyl-be ta-D-ribofuranuronamide derivatives as useful templates for the development of A(2B) adenosine receptor agonists
file con accesso da definire2007 Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli, Romeo; Carrion, Md; Cara, Lcl; Moorman, Ar; Varani, Katia; Borea, Pier Andrea
Synthesis and Biological Evaluation of Novel 2-Amino-3-Aroyl-4-Neopentyl-5-Substituted Thiophene Derivatives as Allosteric Enhancers of the A1 Adenosine Receptor
file con accesso da definire2014 Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Cruz Lopez, O.; Lopez Cara, C.; Kimatrai Salvador, M.; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; Moorman, A. R.; Vincenzi, Fabrizio; Borea, A. P.; Varani, Katia
Synthesis and Biological Evaluation of Novel Allosteric Enhancers of the A1 Adenosine Receptor Based on 2-Amino-3-(4’-Chlorobenzoyl)-4-Substituted-5-Arylethynyl Thiophene
file con accesso da definire2014 Romagnoli, Romeo; Baraldi, Pier Giovanni; A. P., Ijzerman; A., Massink; O., Cruz Lopez; L. C., Lopez Cara; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; A. R., Moorman; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia
Synthesis and biological evaluation of novel N-6-[4-(substituted) sulfonamidophenylcarbamoyl]adenosine-5 '-uronamides as A(3) adenosine receptor agonists
file con accesso da definire2004 Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti, Delia; Bovero, Andrea; DE LAS INFANTAS, Mjp; Moorman, A; Varani, Katia; Borea, Pier Andrea
Synthesis and biological evaluation of novel rhodanine-based structures with antiviral activity towards HHV-6 virus
2022 Gentili, V.; Turrin, G.; Marchetti, P.; Rizzo, S.; Schiuma, G.; Beltrami, S.; Cristofori, V.; Illuminati, D.; Compagnin, G.; Trapella, C.; Rizzo, R.; Bortolotti, D.; Fantinati, A.
Synthesis and biological evaluation of pro-drugs of GW196771, a potent glycine antagonist acting at the NMDA receptor
file con accesso da definire2005 Angusti, A; Durini, Elisa; Vertuani, Silvia; Dalpiaz, Alessandro; Ruffo, A.; DI FABIO, R.; Donati, D.; Pentassuglia, G.; Vitulli, G.; Barnaby, R. J.; Manfredini, Stefano
Synthesis and Biological Evaluation of Pyrazolo[3,4-b]pyridin-4-ones as a New Class of Topoisomerase II Inhibitors
file con accesso da definire2015 AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Prencipe, Filippo; Preti, Delia; Saponaro, Giulia; Romagnoli, Romeo; Gessi, Stefania; Merighi, Stefania; Stefanelli, Angela; Fazzi, Debora; Borea, Pier Andrea; Maia, Rodolfo C. outo; Romeiro, Nelilma C.; Fraga, Carlos A. M; Barreiro, Eliezer J.
Synthesis and biological evaluation of pyrido[2,3-b]pyrazine and pyrido[2,3-b]pyrazine-N-oxide as selective glycine antagonists
file con accesso da definire1996 Cugola, A; Donati, D; Guarneri, M; Micheli, F; Missio, A; Pecunioso, A; Reggiani, A; Tarzia, G; Zanirato, Vinicio
Synthesis and biological evaluation of resveratrol and analogues as apoptosis-inducing agents
file con accesso da definire2003 Roberti, M.; Pizzirani, D.; Simoni, Daniele; Rondanin, Riccardo; Baruchello, Riccardo; Bonora, C.; Buscemi, F.; Grimaudo, S.; Tolomeo, M.
Synthesis and biological evaluation of small anticancer molecules acting as tubulin polymerization inhibitors
2020 Oliva, Paola
Synthesis and biological evaluation of substrate-based inhibitors of 6-phosphogluconate dehydrogenase as potential drugs against African Trypanosomiasis
file con accesso da definire2003 Dardonville, C.; Rinaldi, Eliana; Hanau, Stefania; Barrett, M.; Brun, R.; Gilbert, I. H.
Synthesis and Biological Investigation of Bile Acid-Paclitaxel Hybrids
2022 Melloni, E.; Marchesi, E.; Preti, L.; Casciano, F.; Rimondi, E.; Romani, A.; Secchiero, P.; Navacchia, M. L.; Perrone, D.
Synthesis and biological properties of C-terminal vinyl ketone pseudotripeptides
file con accesso da definire2013 Franceschini, C; Trapella, Claudio; Sforza, F; Gavioli, Riccardo; Marastoni, Mauro
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and Biological Evaluation of Diastereoisomerically Pure N,O-Nucleosides | 2010 | B., Russo; Bortolini, Olga; A., De Nino; A., Garofalo; A., Melicchio; L., Maiuolo | file con accesso da definire |
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity | 2016 | Di Capua, A; Sticozzi, Claudia; Brogi, S; Brindisi, M; Cappelli, A; Sautebin, L; Rossi, A; Pace, ...S; Ghelardini, C; Di Cesare Mannelli, L; Valacchi, Giuseppe; Giorgi, Giulia; Giordani, Alice; Poce, G; Biava, M; Anzini, M. | |
Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents | 2022 | Oliva, Paola; Romagnoli, Romeo; Cacciari, Barbara; Manfredini, Stefano; Padroni, Chiara; Brancale..., Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Milan, Noemi; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta | |
Synthesis and biological evaluation of new 8-heterocyclic xanthine derivative as highly potent and selective human A2B adenosine receptor antagonist | 2006 | Baraldi, Pier Giovanni; Tabrizi, M. A.; Preti, Delia; Bovero, A.; Romagnoli, Romeo; Fruttarolo, F...rancesca; Zaid, N. A.; Moorman, A. R.; Varani, Katia; Gessi, Stefania; Merighi, Stefania; Borea, Pier Andrea | file con accesso da definire |
Synthesis and biological evaluation of new active For-Met-Leu-Phe-OMe analogues containing para-substituted Phe residues. J.Pept.Sci, 18, 418-426, 2012. | 2012 | Mollica, A.; Feliciani, F.; Stefanucci, A.; Costante, R.; Lucente, G.; Pinnen, F.; Notaristefano,... D.; Spisani, Susanna | file con accesso da definire |
Synthesis and biological evaluation of new antitubulin agents containing 2-(30,40,50-trimethoxyanilino)-3,6-disubstituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine Scaffold | 2020 | Romagnoli, Romeo; Prencipe, Filippo; Oliva, Paola; Cacciari, Barbara; Balzarini, Jan; Liekens, Sa...ndra; Hamel, Ernest; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Zurlo, Matteo; Finotti, Alessia; Gambari, Roberto | |
Synthesis and biological evaluation of new vinyl ester pseudotripeptide proteasome inhibitors | 2006 | Marastoni, Mauro; Baldisserotto, Anna; Trapella, Claudio; Gavioli, Riccardo; Tomatis, Roberto | file con accesso da definire |
Synthesis and biological evaluation of novel 1-deoxy-1-[6-[((hetero)arylcarbonyl)hydrazino]-9H-purin-9-yl]-N-ethyl-be ta-D-ribofuranuronamide derivatives as useful templates for the development of A(2B) adenosine receptor agonists | 2007 | Baraldi, Pier Giovanni; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Fruttarolo, Francesca; Romagnoli..., Romeo; Carrion, Md; Cara, Lcl; Moorman, Ar; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Synthesis and Biological Evaluation of Novel 2-Amino-3-Aroyl-4-Neopentyl-5-Substituted Thiophene Derivatives as Allosteric Enhancers of the A1 Adenosine Receptor | 2014 | Romagnoli, Romeo; Baraldi, Pier Giovanni; Carrion, M. D.; Cruz Lopez, O.; Lopez Cara, C.; Kimatra...i Salvador, M.; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; Moorman, A. R.; Vincenzi, Fabrizio; Borea, A. P.; Varani, Katia | file con accesso da definire |
Synthesis and Biological Evaluation of Novel Allosteric Enhancers of the A1 Adenosine Receptor Based on 2-Amino-3-(4’-Chlorobenzoyl)-4-Substituted-5-Arylethynyl Thiophene | 2014 | Romagnoli, Romeo; Baraldi, Pier Giovanni; A. P., Ijzerman; A., Massink; O., Cruz Lopez; L. C., Lo...pez Cara; Saponaro, Giulia; Preti, Delia; AGHAZADEH TABRIZI, Mojgan; Baraldi, Stefania; A. R., Moorman; Vincenzi, Fabrizio; Borea, Pier Andrea; Varani, Katia | file con accesso da definire |
Synthesis and biological evaluation of novel N-6-[4-(substituted) sulfonamidophenylcarbamoyl]adenosine-5 '-uronamides as A(3) adenosine receptor agonists | 2004 | Baraldi, Pier Giovanni; Fruttarolo, Francesca; AGHAZADEH TABRIZI, Mojgan; Romagnoli, Romeo; Preti..., Delia; Bovero, Andrea; DE LAS INFANTAS, Mjp; Moorman, A; Varani, Katia; Borea, Pier Andrea | file con accesso da definire |
Synthesis and biological evaluation of novel rhodanine-based structures with antiviral activity towards HHV-6 virus | 2022 | Gentili, V.; Turrin, G.; Marchetti, P.; Rizzo, S.; Schiuma, G.; Beltrami, S.; Cristofori, V.; Ill...uminati, D.; Compagnin, G.; Trapella, C.; Rizzo, R.; Bortolotti, D.; Fantinati, A. | |
Synthesis and biological evaluation of pro-drugs of GW196771, a potent glycine antagonist acting at the NMDA receptor | 2005 | Angusti, A; Durini, Elisa; Vertuani, Silvia; Dalpiaz, Alessandro; Ruffo, A.; DI FABIO, R.; Donati..., D.; Pentassuglia, G.; Vitulli, G.; Barnaby, R. J.; Manfredini, Stefano | file con accesso da definire |
Synthesis and Biological Evaluation of Pyrazolo[3,4-b]pyridin-4-ones as a New Class of Topoisomerase II Inhibitors | 2015 | AGHAZADEH TABRIZI, Mojgan; Baraldi, Pier Giovanni; Baraldi, Stefania; Prencipe, Filippo; Preti, D...elia; Saponaro, Giulia; Romagnoli, Romeo; Gessi, Stefania; Merighi, Stefania; Stefanelli, Angela; Fazzi, Debora; Borea, Pier Andrea; Maia, Rodolfo C. outo; Romeiro, Nelilma C.; Fraga, Carlos A. M; Barreiro, Eliezer J. | file con accesso da definire |
Synthesis and biological evaluation of pyrido[2,3-b]pyrazine and pyrido[2,3-b]pyrazine-N-oxide as selective glycine antagonists | 1996 | Cugola, A; Donati, D; Guarneri, M; Micheli, F; Missio, A; Pecunioso, A; Reggiani, A; Tarzia, G; Z...anirato, Vinicio | file con accesso da definire |
Synthesis and biological evaluation of resveratrol and analogues as apoptosis-inducing agents | 2003 | Roberti, M.; Pizzirani, D.; Simoni, Daniele; Rondanin, Riccardo; Baruchello, Riccardo; Bonora, C....; Buscemi, F.; Grimaudo, S.; Tolomeo, M. | file con accesso da definire |
Synthesis and biological evaluation of small anticancer molecules acting as tubulin polymerization inhibitors | 2020 | Oliva, Paola | |
Synthesis and biological evaluation of substrate-based inhibitors of 6-phosphogluconate dehydrogenase as potential drugs against African Trypanosomiasis | 2003 | Dardonville, C.; Rinaldi, Eliana; Hanau, Stefania; Barrett, M.; Brun, R.; Gilbert, I. H. | file con accesso da definire |
Synthesis and Biological Investigation of Bile Acid-Paclitaxel Hybrids | 2022 | Melloni, E.; Marchesi, E.; Preti, L.; Casciano, F.; Rimondi, E.; Romani, A.; Secchiero, P.; Navac...chia, M. L.; Perrone, D. | |
Synthesis and biological properties of C-terminal vinyl ketone pseudotripeptides | 2013 | Franceschini, C; Trapella, Claudio; Sforza, F; Gavioli, Riccardo; Marastoni, Mauro | file con accesso da definire |
Legenda icone
- file ad accesso aperto
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile